Shinsuke Inuki

Affiliations

Graduate School of Pharmaceutical Sciences, Kyoto University, Sakyo-ku, Kyoto 606-8501, Japan.

Publications (48)

Scaffold hopping of fused piperidine-type NK3 receptor antagonists to reduce environmental impact.

Bioorganic & medicinal chemistry

Avec: Koki Yamamoto , Shinsuke Inuki , Hiroaki Ohno , Shinya Oishi

Synthesis of Triazolo- and Oxadiazolopiperazines by Gold(I)-Catalyzed Domino Cyclization: Application to the Design of a Mitogen Activated Protein (MAP) Kinase Inhibitor.

Organic letters

Avec: Koki Yamamoto , Yasushi Yoshikawa , Masahito Ohue , Shinsuke Inuki , Hiroaki Ohno , Shinya Oishi

Total Synthesis of Zephycarinatines via Photocatalytic Reductive Radical ipso-Cyclization.

Angewandte Chemie (International ed. in English)

Avec: Haruka Takeuchi , Shinsuke Inuki , Kohei Nakagawa , Takaaki Kawabe , Atsuhiko Ichimura , Shinya Oishi , Hiroaki Ohno

Structure-activity relationship studies of tetrahydroquinolone derivatives as GPR41 modulators.

Bioorganic & medicinal chemistry letters

Avec: Shinsuke Inuki , Junki Miyamoto , Naoki Hashimoto , Hidenori Shimizu , Hitomi Tabuchi , Atsuko Kawai , Luca C Greiner , Ikuo Kimura , Hiroaki Ohno

[Elucidation of Biological Mechanisms Using Synthetic Natural Products and Their Derivatives].

Yakugaku zasshi : Journal of the Pharmaceutical Society of Japan

Avec: Shinsuke Inuki

Construction of the Pyrrolo[2,3-

The Journal of organic chemistry

Avec: Junpei Matsuoka , Hiroshi Kumagai , Shinsuke Inuki , Shinya Oishi , Hiroaki Ohno

Novel anti-flavivirus drugs targeting the nucleolar distribution of core protein.

Virology

Avec: Makoto Tokunaga , Yoichi Miyamoto , Tatsuya Suzuki , Mayumi Otani , Shinsuke Inuki , Tsuyoshi Esaki , Chioko Nagao , Kenji Mizuguchi , Hiroaki Ohno , Yoshihiro Yoneda , Toru Okamoto , Masahiro Oka , Yoshiharu Matsuura

The effects of 5-OP-RU stereochemistry on its stability and MAIT-MR1 axis.

Chembiochem : a European journal of chemical biology

Avec: Takuro Matsuoka , Chihiro Motozono , Akira Hattori , Hideaki Kakeya , Sho Yamasaki , Shinya Oishi , Hiroaki Ohno , Shinsuke Inuki

Gold(I)-Catalyzed Cascade Cyclization of Alkynyl Indoles for the Stereoselective Construction of the Quaternary Carbon Center of Akuammiline Alkaloids.

The Journal of organic chemistry

Avec: Naoki Hashimoto , Junichi Taguchi , Norihito Arichi , Shinsuke Inuki , Hiroaki Ohno

Gold(I)-Catalyzed Bis-Cyclization of Allenynes for the Synthesis of Strained and Planar Polycyclic Compounds.

Angewandte Chemie (International ed. in English)

Avec: Hitomi Tsuno , Jingfeng Shen , Hiroki Komatsu , Norihito Arichi , Shinsuke Inuki , Hiroaki Ohno

Chemical Synthesis and Molecular Interaction Analysis of α-Galactosyl Ceramide Derivatives as CD1d Ligands.

Methods in molecular biology (Clifton, N.J.)

Avec: Kazunari Ueki , Kodai Sueyoshi , Shinsuke Inuki , Yukari Fujimoto

Synthesis of the full-length hepatitis B virus core protein and its capsid formation.

Organic & biomolecular chemistry

Avec: Keisuke Aoki , Shugo Tsuda , Naoko Ogata , Michiyo Kataoka , Jumpei Sasaki , Shinsuke Inuki , Hiroaki Ohno , Koichi Watashi , Taku Yoshiya , Shinya Oishi

Synthesis of labionin and avionin precursors

Organic & biomolecular chemistry

Avec: Ayuta Yamaguchi , Naoki Obiya , Norihito Arichi , Shinya Oishi , Hiroaki Ohno , Shinsuke Inuki

Polar functional group-containing glycolipid CD1d ligands modulate cytokine-biasing responses and prevent experimental colitis.

Scientific reports

Avec: Shinsuke Inuki , Natsumi Hirata , Emi Kashiwabara , Junichiro Kishi , Toshihiko Aiba , Toshiaki Teratani , Wataru Nakamura , Yoshimi Kojima , Toru Maruyama , Takanori Kanai , Yukari Fujimoto

Construction of Quaternary Carbon Stereocenter of α-Tertiary Amine through Remote C-H Functionalization of Tris Derivatives: Enantioselective Total Synthesis of Myriocin.

Organic letters

Avec: Takashi Miyagawa , Shinsuke Inuki , Shinya Oishi , Hiroaki Ohno

Structure-activity relationship studies of Bz amide-containing α-GalCer derivatives as natural killer T cell modulators.

Bioorganic & medicinal chemistry letters

Avec: Junichiro Kishi , Shinsuke Inuki , Natsumi Hirata , Emi Kashiwabara , Daisuke Yoshidome , Osamu Ichihara , Yukari Fujimoto

Design and Discovery of Covalent α-GalCer Derivatives as Potent CD1d Ligands.

ACS chemical biology

Avec: Junichiro Kishi , Shinsuke Inuki , Emi Kashiwabara , Takehiro Suzuki , Naoshi Dohmae , Yukari Fujimoto

Total Synthesis of Dictyodendrins A-F by the Gold-Catalyzed Cascade Cyclization of Conjugated Diyne with Pyrrole.

Chemistry (Weinheim an der Bergstrasse, Germany)

Avec: Junpei Matsuoka , Shinsuke Inuki , Yuka Matsuda , Yoichi Miyamoto , Mayumi Otani , Masahiro Oka , Shinya Oishi , Hiroaki Ohno

Engineering a Low-Immunogenic Mirror-Image VHH against Vascular Endothelial Growth Factor.

ACS chemical biology

Avec: Keisuke Aoki , Katsuaki Higashi , Sakiho Oda , Asako Manabe , Kayuu Maeda , Jyoji Morise , Shogo Oka , Shinsuke Inuki , Hiroaki Ohno , Shinya Oishi , Motohiro Nonaka

Chemical Synthesis and Evaluation of Exopolysaccharide Fragments Produced by Leuconostoc mesenteroides Strain NTM048.

Chemical & pharmaceutical bulletin

Avec: Shinsuke Inuki , Hitomi Tabuchi , Chiaki Matsuzaki , Yasunori Yonejima , Keiko Hisa , Ikuo Kimura , Kenji Yamamoto , Hiroaki Ohno

Design of Synthetic Surrogates for the Macrolactone Linker Motif in Coibamide A.

ACS medicinal chemistry letters

Avec: Rikito Suzuki , Daphne R Mattos , Takashi Kitamura , Rina Tsujioka , Kazuya Kobayashi , Shinsuke Inuki , Hiroaki Ohno , Jane E Ishmael , Kerry L McPhail , Shinya Oishi

Design and Synthesis of Monobody Variants with Low Immunogenicity.

ACS medicinal chemistry letters

Avec: Naoya Iwamoto , Yukino Sato , Asako Manabe , Shinsuke Inuki , Hiroaki Ohno , Motohiro Nonaka , Shinya Oishi

Synthetic Studies on FNC-RED and Its Analogues Containing an All

The Journal of organic chemistry

Avec: Shinsuke Inuki , Keisuke Sato , Naoto Zui , Ryosuke Yamaguchi , Takanori Matsumaru , Yukari Fujimoto

Nonbiomimetic total synthesis of indole alkaloids using alkyne-based strategies.

Organic & biomolecular chemistry

Avec: Hiroaki Ohno , Shinsuke Inuki

Construction of Tricyclic Nitrogen Heterocycles by a Gold(I)-Catalyzed Cascade Cyclization of Allenynes and Application to Polycyclic π-Electron Systems.

Angewandte Chemie (International ed. in English)

Avec: Hiroki Komatsu , Takaya Ikeuchi , Hitomi Tsuno , Norihito Arichi , Kosuke Yasui , Shinya Oishi , Shinsuke Inuki , Aiko Fukazawa , Hiroaki Ohno

Access to Indole-Fused Benzannulated Medium-Sized Rings through a Gold(I)-Catalyzed Cascade Cyclization of Azido-Alkynes.

Chemistry (Weinheim an der Bergstrasse, Germany)

Avec: Luca C Greiner , Shinsuke Inuki , Norihito Arichi , Shinya Oishi , Rikito Suzuki , Tomohiro Iwai , Masaya Sawamura , A Stephen K Hashmi , Hiroaki Ohno

Design of Coibamide A Mimetics with Improved Cellular Bioactivity.

ACS medicinal chemistry letters

Avec: Takashi Kitamura , Rikito Suzuki , Shinsuke Inuki , Hiroaki Ohno , Kerry L McPhail , Shinya Oishi

Gold(I)-Catalyzed Benzylic C(sp

Angewandte Chemie (International ed. in English)

Avec: Luca C Greiner , Norihito Arichi , Shinsuke Inuki , Hiroaki Ohno

Discovery of Bis-sulfonamides as Novel Inhibitors of Mitochondrial NADH-Quinone Oxidoreductase (Complex I).

ACS medicinal chemistry letters

Avec: Atsuhito Tsuji , Takahiro Masuya , Norihito Arichi , Shinsuke Inuki , Masatoshi Murai , Hideto Miyoshi , Hiroaki Ohno

Establishment of an MR1 Presentation Reporter Screening System and Identification of Phenylpropanoid Derivatives as MR1 Ligands.

Journal of medicinal chemistry

Avec: Takuro Matsuoka , Akira Hattori , Shinya Oishi , Mitsugu Araki , Biao Ma , Toshiki Fujii , Norihito Arichi , Yasushi Okuno , Hideaki Kakeya , Sho Yamasaki , Hiroaki Ohno , Shinsuke Inuki

Mirror-Image Single-Domain Antibody for a Novel Nonimmunogenic Drug Scaffold.

Bioconjugate chemistry

Avec: Keisuke Aoki , Asako Manabe , Hiroyuki Kimura , Yohei Katoh , Shinsuke Inuki , Hiroaki Ohno , Motohiro Nonaka , Shinya Oishi

Sulfated bile acid is a host-derived ligand for MAIT cells.

Science immunology

Avec: Emi Ito , Shinsuke Inuki , Yoshihiro Izumi , Masatomo Takahashi , Yuki Dambayashi , Lisa Ciacchi , Wael Awad , Ami Takeyama , Kensuke Shibata , Shotaro Mori , Jeffrey Y W Mak , David P Fairlie , Takeshi Bamba , Eri Ishikawa , Masamichi Nagae , Jamie Rossjohn , Sho Yamasaki

Synthesis of Sulfilimines via Visible-Light-Mediated Triplet Energy Transfer to Sulfonyl Azides.

Chemistry (Weinheim an der Bergstrasse, Germany)

Avec: Norihito Arichi , Tsuyoshi Amano , Shuhan Wu , Shinsuke Inuki , Hiroaki Ohno

Development of Ribityllumazine Analogue as Mucosal-Associated Invariant T Cell Ligands.

Journal of the American Chemical Society

Avec: Ryosuke Takasaki , Emi Ito , Masamichi Nagae , Yuki Takahashi , Takuro Matsuoka , Wakana Yasue , Norihito Arichi , Hiroaki Ohno , Sho Yamasaki , Shinsuke Inuki

Total Synthesis of Dictyodendrins A-F by the Gold-Catalyzed Cascade Cyclization of Conjugated Diyne with Pyrrole.

Chemistry (Weinheim an der Bergstrasse, Germany)

Avec: Junpei Matsuoka , Shinsuke Inuki , Yuka Matsuda , Yoichi Miyamoto , Mayumi Otani , Masahiro Oka , Shinya Oishi , Hiroaki Ohno

Total Synthesis of (+)-Polyoxamic Acid via Visible-Light-Mediated Photocatalytic β-Scission and 1,5-Hydrogen Atom Transfer of Glucose Derivative.

The Journal of organic chemistry

Avec: Takuro Matsuoka , Shinsuke Inuki , Takashi Miyagawa , Shinya Oishi , Hiroaki Ohno

Gold(I)-Catalyzed Cascade Cyclization of Anilines with Diynes: Controllable Formation of Eight-Membered Ring-Fused Indoles and Propellane-Type Indolines.

The Journal of organic chemistry

Avec: Ayuta Yamaguchi , Shinsuke Inuki , Yusuke Tokimizu , Shinya Oishi , Hiroaki Ohno

Gold(I)-Catalyzed Cascade Cyclization Reactions of Allenynes for the Synthesis of Fused Cyclopropanes and Acenaphthenes.

Angewandte Chemie (International ed. in English)

Avec: Takaya Ikeuchi , Shinsuke Inuki , Shinya Oishi , Hiroaki Ohno

Azido-Alkynes in Gold(I)-Catalyzed Indole Syntheses.

Chemical record (New York, N.Y.)

Avec: Luca C Greiner , Junpei Matsuoka , Shinsuke Inuki , Hiroaki Ohno

Access to Indole-Fused Benzannulated Medium-Sized Rings through a Gold(I)-Catalyzed Cascade Cyclization of Azido-Alkynes.

Chemistry (Weinheim an der Bergstrasse, Germany)

Avec: Luca C Greiner , Shinsuke Inuki , Norihito Arichi , Shinya Oishi , Rikito Suzuki , Tomohiro Iwai , Masaya Sawamura , A Stephen K Hashmi , Hiroaki Ohno

Synthetic studies on the extracellular domain of the T cell immunoreceptor with immunoglobulin and immunoreceptor tyrosine-based inhibitory motif domain (TIGIT) using Trt-K

Bioorganic & medicinal chemistry

Avec: Naoya Iwamoto , Jumpei Sasaki , Saya Ohno , Keisuke Aoki , Yusuke Usui , Shinsuke Inuki , Hiroaki Ohno , Shinya Oishi

Variational autoencoder-based chemical latent space for large molecular structures with 3D complexity.

Communications chemistry

Avec: Toshiki Ochiai , Tensei Inukai , Manato Akiyama , Kairi Furui , Masahito Ohue , Nobuaki Matsumori , Shinsuke Inuki , Motonari Uesugi , Toshiaki Sunazuka , Kazuya Kikuchi , Hideaki Kakeya , Yasubumi Sakakibara

Construction of a Bicyclo[2.2.2]octene Skeleton via a Visible-Light-Mediated Radical Cascade Reaction of Amino Acid Derivatives with

Organic letters

Avec: Yuki Yoshida , Haruka Takeuchi , Kohei Nakagawa , Toshiki Fujii , Norihito Arichi , Shinya Oishi , Hiroaki Ohno , Shinsuke Inuki

Archaeal Glycerolipids Are Recognized by C-Type Lectin Receptor Mincle.

Journal of the American Chemical Society

Avec: Shiori Oka , Miyuki Watanabe , Emi Ito , Ami Takeyama , Takuro Matsuoka , Masatomo Takahashi , Yoshihiro Izumi , Norihito Arichi , Hiroaki Ohno , Sho Yamasaki , Shinsuke Inuki

Mirror-Image Human Serum Albumin Domain III as a Tool for Analyzing Site II-Dependent Molecular Recognition.

Bioconjugate chemistry

Avec: Naoya Iwamoto , Takuma Kai , Shinsuke Inuki , Hiroaki Ohno , Hitoshi Maeda , Hiroshi Watanabe , Toru Maruyama , Shinya Oishi

Construction of the Akuammiline Alkaloid Core Structure via Stereoselective E-Ring Formation.

The Journal of organic chemistry

Avec: Naoki Hashimoto , Junichi Taguchi , Takumi Kasagi , Norihito Arichi , Shinsuke Inuki , Hiroaki Ohno

The identification of novel small extracellular vesicle (sEV) production modulators using luciferase-based sEV quantification method.

Journal of extracellular biology

Avec: Aki Yamamoto , Yuki Takahashi , Shinsuke Inuki , Shumpei Nakagawa , Kodai Nakao , Hiroaki Ohno , Masao Doi , Yoshinobu Takakura

Chemical Synthesis of Interleukin-6 for Mirror-Image Screening.

Bioconjugate chemistry

Avec: Keisuke Aoki , Kayuu Maeda , Shinsuke Inuki , Hiroaki Ohno , Motohiro Nonaka , Shinya Oishi

Réseau de co-auteurs

Hiroaki Ohno 40 collaborations

Shinya Oishi 26 collaborations

Norihito Arichi 14 collaborations

Luca C Greiner 5 collaborations

Takuro Matsuoka 5 collaborations

Sho Yamasaki 5 collaborations

Yukari Fujimoto 5 collaborations

Keisuke Aoki 5 collaborations

Junpei Matsuoka 4 collaborations

Motohiro Nonaka 4 collaborations

Rikito Suzuki 4 collaborations

Naoki Hashimoto 3 collaborations

Yoichi Miyamoto 3 collaborations

Mayumi Otani 3 collaborations

Masahiro Oka 3 collaborations

Hideaki Kakeya 3 collaborations

Emi Kashiwabara 3 collaborations

Junichiro Kishi 3 collaborations

Asako Manabe 3 collaborations

Naoya Iwamoto 3 collaborations

Emi Ito 3 collaborations

Koki Yamamoto 2 collaborations

Masahito Ohue 2 collaborations

Haruka Takeuchi 2 collaborations

Kohei Nakagawa 2 collaborations

Hitomi Tabuchi 2 collaborations

Ikuo Kimura 2 collaborations

Akira Hattori 2 collaborations

Junichi Taguchi 2 collaborations

Hitomi Tsuno 2 collaborations

Hiroki Komatsu 2 collaborations

Jumpei Sasaki 2 collaborations

Ayuta Yamaguchi 2 collaborations

Natsumi Hirata 2 collaborations

Toru Maruyama 2 collaborations

Takashi Miyagawa 2 collaborations

Yuka Matsuda 2 collaborations

Kayuu Maeda 2 collaborations

Takashi Kitamura 2 collaborations

Kerry L McPhail 2 collaborations

Takaya Ikeuchi 2 collaborations

Tomohiro Iwai 2 collaborations

Masaya Sawamura 2 collaborations

A Stephen K Hashmi 2 collaborations

Toshiki Fujii 2 collaborations

Yoshihiro Izumi 2 collaborations

Masatomo Takahashi 2 collaborations

Ami Takeyama 2 collaborations

Masamichi Nagae 2 collaborations

Yuki Takahashi 2 collaborations

Yasushi Yoshikawa 1 collaboration

Takaaki Kawabe 1 collaboration

Atsuhiko Ichimura 1 collaboration

Junki Miyamoto 1 collaboration

Hidenori Shimizu 1 collaboration

Atsuko Kawai 1 collaboration

Hiroshi Kumagai 1 collaboration

Makoto Tokunaga 1 collaboration

Tatsuya Suzuki 1 collaboration

Tsuyoshi Esaki 1 collaboration

Chioko Nagao 1 collaboration

Kenji Mizuguchi 1 collaboration

Yoshihiro Yoneda 1 collaboration

Toru Okamoto 1 collaboration

Yoshiharu Matsuura 1 collaboration

Chihiro Motozono 1 collaboration

Jingfeng Shen 1 collaboration

Kazunari Ueki 1 collaboration

Kodai Sueyoshi 1 collaboration

Shugo Tsuda 1 collaboration

Naoko Ogata 1 collaboration

Michiyo Kataoka 1 collaboration

Koichi Watashi 1 collaboration

Taku Yoshiya 1 collaboration

Naoki Obiya 1 collaboration

Toshihiko Aiba 1 collaboration

Toshiaki Teratani 1 collaboration

Wataru Nakamura 1 collaboration

Yoshimi Kojima 1 collaboration

Takanori Kanai 1 collaboration

Daisuke Yoshidome 1 collaboration

Osamu Ichihara 1 collaboration

Takehiro Suzuki 1 collaboration

Naoshi Dohmae 1 collaboration

Katsuaki Higashi 1 collaboration

Sakiho Oda 1 collaboration

Jyoji Morise 1 collaboration

Shogo Oka 1 collaboration

Chiaki Matsuzaki 1 collaboration

Yasunori Yonejima 1 collaboration

Keiko Hisa 1 collaboration

Kenji Yamamoto 1 collaboration

Daphne R Mattos 1 collaboration

Rina Tsujioka 1 collaboration

Kazuya Kobayashi 1 collaboration

Jane E Ishmael 1 collaboration

Yukino Sato 1 collaboration

Keisuke Sato 1 collaboration

Naoto Zui 1 collaboration

Ryosuke Yamaguchi 1 collaboration

Takanori Matsumaru 1 collaboration

Kosuke Yasui 1 collaboration

Aiko Fukazawa 1 collaboration

Atsuhito Tsuji 1 collaboration

Takahiro Masuya 1 collaboration

Masatoshi Murai 1 collaboration

Hideto Miyoshi 1 collaboration

Mitsugu Araki 1 collaboration

Biao Ma 1 collaboration

Yasushi Okuno 1 collaboration

Hiroyuki Kimura 1 collaboration

Yohei Katoh 1 collaboration

Yuki Dambayashi 1 collaboration

Lisa Ciacchi 1 collaboration

Wael Awad 1 collaboration

Kensuke Shibata 1 collaboration

Shotaro Mori 1 collaboration

Jeffrey Y W Mak 1 collaboration

David P Fairlie 1 collaboration

Takeshi Bamba 1 collaboration

Eri Ishikawa 1 collaboration

Jamie Rossjohn 1 collaboration

Tsuyoshi Amano 1 collaboration

Shuhan Wu 1 collaboration

Ryosuke Takasaki 1 collaboration

Wakana Yasue 1 collaboration

Yusuke Tokimizu 1 collaboration

Saya Ohno 1 collaboration

Yusuke Usui 1 collaboration

Toshiki Ochiai 1 collaboration

Tensei Inukai 1 collaboration

Manato Akiyama 1 collaboration

Kairi Furui 1 collaboration

Nobuaki Matsumori 1 collaboration

Motonari Uesugi 1 collaboration

Toshiaki Sunazuka 1 collaboration

Kazuya Kikuchi 1 collaboration

Yasubumi Sakakibara 1 collaboration

Yuki Yoshida 1 collaboration

Shiori Oka 1 collaboration

Miyuki Watanabe 1 collaboration

Takuma Kai 1 collaboration

Hitoshi Maeda 1 collaboration

Hiroshi Watanabe 1 collaboration

Takumi Kasagi 1 collaboration

Aki Yamamoto 1 collaboration

Shumpei Nakagawa 1 collaboration

Kodai Nakao 1 collaboration

Masao Doi 1 collaboration

Yoshinobu Takakura 1 collaboration