Dante Rotili

Affiliations
  • Dipartimento di Chimica e Tecnologie del Farmaco , "Sapienza" Università di Roma , 00185 Rome , Italy.

Publications (66)

Structure-Reactivity Relationships on Substrates and Inhibitors of the Lysine Deacylase Sirtuin 2 from

Journal of medicinal chemistry
Avec: Daria Monaldi , Julien Lancelot , Martin Marek , Nathalie Wössner , Alessia Lucidi , Daniela Tomaselli , Elizabeth Ramos-Morales , Christophe Romier , Raymond J Pierce , Antonello Mai , Manfred Jung

Identification of novel quinazoline derivatives as potent antiplasmodial agents.

European journal of medicinal chemistry
Avec: Anne Bouchut , Christine Pierrot , Sergio Valente , Sophia Lafitte , Johan Schultz , Urban Hoglund , Roberta Mazzone , Alessia Lucidi , Giancarlo Fabrizi , Dany Pechalrieu , Paola B Arimondo , Tina S Skinner-Adams , Ming Jang Chua , Kathy T Andrews , Antonello Mai , Jamal Khalife

Lysine Acetyltransferase Inhibitors From Natural Sources.

Frontiers in pharmacology
Avec: Francesco Fiorentino , Antonello Mai ,

Inhibition of Histone Demethylases LSD1 and UTX Regulates ERα Signaling in Breast Cancer.

Cancers
Avec: Rosaria Benedetti , Carmela Dell'Aversana , Tommaso De Marchi , Ning Qing Liu , Boris Novakovic , Serena Boccella , Salvatore Di Maro , Sandro Cosconati , Alfonso Baldi , Emma Niméus , Johan Schultz , Urban Höglund , Sabatino Maione , Chiara Papulino , Ugo Chianese , Francesco Iovino , Antonio Federico , Antonello Mai , Hendrik G Stunnenberg , Angela Nebbioso , Lucia Altucci

Targeting histone acetylation/deacetylation in parasites: an update (2017-2020).

Current opinion in chemical biology
Avec: Rossella Fioravanti , Nicola Mautone , Annarita Rovere , Antonello Mai

Emerging Therapeutic Potential of SIRT6 Modulators.

Journal of medicinal chemistry
Avec: Francesco Fiorentino , Antonello Mai ,

Metabolic Rewiring by Loss of Sirt5 Promotes Kras-Induced Pancreatic Cancer Progression.

Gastroenterology
Avec: Tuo Hu , Surendra K Shukla , Enza Vernucci , Chunbo He , Dezhen Wang , Ryan J King , Kanupriya Jha , Kasturi Siddhanta , Nicholas J Mullen , Kuldeep S Attri , Divya Murthy , Nina V Chaika , Ravi Thakur , Scott E Mulder , Camila G Pacheco , Xiao Fu , Robin R High , Fang Yu , Audrey Lazenby , Clemens Steegborn , Ping Lan , Kamiya Mehla , Sarika Chaudhary , Sergio Valente , Marco Tafani , Antonello Mai , Johan Auwerx , Eric Verdin , David Tuveson , Pankaj K Singh

The Nitrobenzoxadiazole Derivative NBDHEX Behaves as

Pharmaceuticals (Basel, Switzerland)
Avec: Giulia Siciliano , Veronica Di Paolo , Rossella Migale , Francesca Pedini , Marialuisa Casella , Serena Camerini , Daniele Dalzoppo , Rob Henderson , Tonnie Huijs , Koen J Dechering , Antonello Mai , Anna Maria Caccuri , Marco Lalle , Luigi Quintieri , Pietro Alano

Biochemical Functions and Clinical Characterizations of the Sirtuins in Diabetes-Induced Retinal Pathologies.

International journal of molecular sciences
Avec: Samanta Taurone , Chiara De Ponte , Elena De Santis , Antonello Mai , Francesco Fiorentino , Susanna Scarpa , Marco Artico , Alessandra Micera

The α-tubulin acetyltransferase ATAT1: structure, cellular functions, and its emerging role in human diseases.

Cellular and molecular life sciences : CMLS
Avec: Angela Iuzzolino , Francesca Romana Pellegrini , Francesca Degrassi , Daniela Trisciuoglio

Emerging Roles of SIRT5 in Metabolism, Cancer, and SARS-CoV-2 Infection.

Cells
Avec: Emanuele Fabbrizi , Francesco Fiorentino , Vincenzo Carafa , Lucia Altucci , Antonello Mai ,

Epigenetic polypharmacology: A new frontier for epi-drug discovery.

Medicinal research reviews
Avec: Daniela Tomaselli , Alessia Lucidi , Antonello Mai

Comparison of the effects of synthetic and plant-derived mTOR regulators on healthy human ovarian cells.

European journal of pharmacology
Avec: Alexander V Sirotkin , Erika Adamcova , Antonello Mai , Milos Mlyncek , Lamjed Mansour , Saleh Alwasel , Abdel Halim Harrath

Histone deacetylase inhibitors exert anti-tumor effects on human adherent and stem-like glioma cells.

Clinical epigenetics
Avec: Halina Was , Sylwia K Krol , Antonello Mai , Bartosz Wojtas , Bozena Kaminska , Marta Maleszewska

Sirtuin modulators: where are we now? A review of patents from 2015 to 2019.

Expert opinion on therapeutic patents
Avec: Nicola Mautone , Clemens Zwergel , Antonello Mai ,

Recent advances in epigenetic proteolysis targeting chimeras (Epi-PROTACs).

European journal of medicinal chemistry
Avec: Daniela Tomaselli , Nicola Mautone , Antonello Mai ,

First-in-Class Inhibitors of the Ribosomal Oxygenase MINA53.

Journal of medicinal chemistry
Avec: Radosław P Nowak , Anthony Tumber , Eline Hendrix , Mohammad Salik Zeya Ansari , Manuela Sabatino , Lorenzo Antonini , Regina Andrijes , Eidarus Salah , Nicola Mautone , Francesca Romana Pellegrini , Klemensas Simelis , Akane Kawamura , Catrine Johansson , Daniela Passeri , Roberto Pellicciari , Alessia Ciogli , Donatella Del Bufalo , Rino Ragno , Mathew L Coleman , Daniela Trisciuoglio , Antonello Mai , Udo Oppermann , Christopher J Schofield ,

Mass spectrometry enables the discovery of inhibitors of an LPS transport assembly

Chemical communications (Cambridge, England)
Avec: Francesco Fiorentino , Antonello Mai , Jani R Bolla , Carol V Robinson

Sirtuin modulators: past, present, and future perspectives.

Future medicinal chemistry
Avec: Francesco Fiorentino , Nicola Mautone , Martina Menna , Francesca D'Acunzo , Antonello Mai ,

Successes and challenges in the development of BD1-selective BET inhibitors: a patent review.

Expert opinion on therapeutic patents
Avec: Monica Viviano , Alessandra Cipriano , Emanuele Fabbrizi , Alessandra Feoli , Sabrina Castellano , Gianluca Sbardella , Antonello Mai , Ciro Milite ,

(Heteroarylmethyl)benzoic Acids as a New Class of Bacterial Cystathionine γ-Lyase Inhibitors: Synthesis, Biological Evaluation, and Molecular Modeling.

ACS infectious diseases
Avec: Anastasia Golovina , Eleonora Proia , Francesco Fiorentino , Maxim Yunin , Maria Kasatkina , Nailya Zigangirova , Anna Soloveva , Elena Sysolyatina , Svetlana Ermolaeva , Roman Novikov , Sergei Silonov , Sergei Pushkin , Milan Mladenović , Julia Isakova , Albina Belik , Maxim Nawrozkij , Rino Ragno , Roman Ivanov

Histone lysine demethylase inhibition reprograms prostate cancer metabolism and mechanics.

Molecular metabolism
Avec: Ugo Chianese , Chiara Papulino , Eugenia Passaro , Tom Mj Evers , Mehrad Babaei , Antonella Toraldo , Tommaso De Marchi , Emma Niméus , Vincenzo Carafa , Maria Maddalena Nicoletti , Nunzio Del Gaudio , Nunzia Iaccarino , Antonio Randazzo , Antonello Mai , Salvatore Cappabianca , Alireza Mashaghi , Fortunato Ciardiello , Lucia Altucci , Rosaria Benedetti

Systematic Design of Adenosine Analogs as Inhibitors of a

Journal of medicinal chemistry
Avec: Jujun Zhou , John R Horton , Martina Menna , Francesco Fiorentino , Ren Ren , Dan Yu , Taraneh Hajian , Masoud Vedadi , Giulia Mazzoccanti , Alessia Ciogli , Elmar Weinhold , Michael Hüben , Robert M Blumenthal , Xing Zhang , Antonello Mai , Xiaodong Cheng

Antihistamines, phenothiazine-based antipsychotics, and tricyclic antidepressants potently activate pharmacologically relevant human carbonic anhydrase isoforms II and VII.

Journal of enzyme inhibition and medicinal chemistry
Avec: Francesco Fiorentino , Alessio Nocentini , Claudiu T Supuran , Antonello Mai

The Pan-Sirtuin Inhibitor MC2494 Regulates Mitochondrial Function in a Leukemia Cell Line.

Frontiers in oncology
Avec: Vincenzo Carafa , Rosita Russo , Laura Della Torre , Francesca Cuomo , Carmela Dell'Aversana , Federica Sarno , Giulia Sgueglia , Marzia Di Donato , Antonello Mai , Angela Nebbioso , Gilda Cobellis , Angela Chambery , Lucia Altucci

Pharmacological inhibition of lysine-specific demethylase 1 (LSD1) induces global transcriptional deregulation and ultrastructural alterations that impair viability in Schistosoma mansoni.

PLoS neglected tropical diseases
Avec: Vitor Coutinho Carneiro , Isabel Caetano de Abreu da Silva , Murilo Sena Amaral , Adriana S A Pereira , Gilbert Oliveira Silveira , David da Silva Pires , Sergio Verjovski-Almeida , Frank J Dekker , Antonello Mai , Eduardo José Lopes-Torres , Dina Robaa , Wolfgang Sippl , Raymond J Pierce , M Teresa Borrello , A Ganesan , Julien Lancelot , Silvana Thiengo , Monica Ammon Fernandez , Amanda Roberta Revoredo Vicentino , Marina Moraes Mourão , Fernanda Sales Coelho , Marcelo Rosado Fantappié

Multimodal evaluation of

Physica medica : PM : an international journal devoted to the applications of physics to medicine and biology : official journal of the Italian Association of Biomedical Physics (AIFB)
Avec: Andrea Ciardiello , Saverio Altieri , Francesca Ballarini , Valerio Bocci , Silva Bortolussi , Laura Cansolino , Daniele Carlotti , Mario Ciocca , Riccardo Faccini , Angelica Facoetti , Cinzia Ferrari , Luca Ficcadenti , Emiliano Furfaro , Stefano Giagu , Francesco Iacoangeli , Giampiero Macioce , Carlo Mancini-Terracciano , Andrea Messina , Luisa Milazzo , Severina Pacifico , Simona Piccolella , Ian Postuma , Valerio Vercesi , Cecilia Voena , Francesca Vulcano , Silvia Capuani

Regulatory Interplay between miR-181a-5p and Estrogen Receptor Signaling Cascade in Breast Cancer.

Cancers
Avec: Rosaria Benedetti , Chiara Papulino , Giulia Sgueglia , Ugo Chianese , Tommaso De Marchi , Francesco Iovino , Antonello Mai , Emma Niméus , Carmela Dell' Aversana , Lucia Altucci

Novel non-covalent LSD1 inhibitors endowed with anticancer effects in leukemia and solid tumor cellular models.

European journal of medicinal chemistry
Avec: Martina Menna , Francesco Fiorentino , Biagina Marrocco , Alessia Lucidi , Stefano Tomassi , Domenica Cilli , Mauro Romanenghi , Matteo Cassandri , Silvia Pomella , Michele Pezzella , Donatella Del Bufalo , Mohammad Salik Zeya Ansari , Nevena Tomašević , Milan Mladenović , Monica Viviano , Gianluca Sbardella , Rossella Rota , Daniela Trisciuoglio , Saverio Minucci , Andrea Mattevi , Antonello Mai

Molecular insights into RmcA-mediated c-di-GMP consumption: Linking redox potential to biofilm morphogenesis in Pseudomonas aeruginosa.

Microbiological research
Avec: Chiara Scribani Rossi , Kelly Eckartt , Elisabetta Scarchilli , Simone Angeli , Alexa Price-Whelan , Adele Di Matteo , Maelenn Chevreuil , Bertrand Raynal , Alessandro Arcovito , Noah Giacon , Francesco Fiorentino , Antonello Mai , Manuel Espinosa-Urgel , Francesca Cutruzzolà , Lars E P Dietrich , Alessio Paone , Alessandro Paiardini , Serena Rinaldo

SIRT6 Protects Against Lipopolysaccharide-Induced Inflammation in Human Pulmonary Lung Microvascular Endothelial Cells.

Inflammation
Avec: Jinping Wang , Jinque Luo , Antonello Mai , Clemens Steegborn , Suowen Xu , Zheng Gen Jin

Role of SIRT3 in Microgravity Response: A New Player in Muscle Tissue Recovery.

Cells
Avec: Michele Aventaggiato , Federica Barreca , Laura Vitiello , Simone Vespa , Sergio Valente , Antonello Mai , Lavinia Vittoria Lotti , Luigi Sansone , Matteo A Russo , Mariano Bizzarri , Elisabetta Ferretti , Marco Tafani

Quinoline-based compounds can inhibit diverse enzymes that act on DNA.

bioRxiv : the preprint server for biology
Avec: Jujun Zhou , Qin Chen , Ren Ren , Jie Yang , Bigang Liu , John R Horton , Caleb Chang , Chuxuan Li , Leora Maksoud , Yifei Yang , Xing Zhang , Robert M Blumenthal , Taiping Chen , Yang Gao , Sergio Valente , Antonello Mai , Xiaodong Cheng

Activation and inhibition of sirtuins: From bench to bedside.

Medicinal research reviews
Avec: Francesco Fiorentino , Emanuele Fabbrizi , Antonello Mai ,

Transmission-Blocking Strategies for Malaria Eradication: Recent Advances in Small-Molecule Drug Development.

Pharmaceuticals (Basel, Switzerland)
Avec: Federico Appetecchia , Emanuele Fabbrizi , Francesco Fiorentino , Sara Consalvi , Mariangela Biava , Giovanna Poce ,

Prognostic Impact of H19/Cell Adhesion Molecules Circuitry on Prostate Cancer Biopsy.

Biomedicines
Avec: Valeria Pecci , Francesco Pierconti , Angela Carlino , Francesco Pinto , Ugo Gradilone , Sara De Martino , Claudio Grassi , Alfredo Pontecorvi , Carlo Gaetano , Lidia Strigari , Antonella Farsetti , Simona Nanni

Quinoline-based compounds can inhibit diverse enzymes that act on DNA.

Cell chemical biology
Avec: Jujun Zhou , Qin Chen , Ren Ren , Jie Yang , Bigang Liu , John R Horton , Caleb Chang , Chuxuan Li , Leora Maksoud , Yifei Yang , Abhinav K Jain , Xing Zhang , Robert M Blumenthal , Taiping Chen , Yang Gao , Sergio Valente , Antonello Mai , Xiaodong Cheng

Sirt4: A Multifaceted Enzyme at the Crossroads of Mitochondrial Metabolism and Cancer.

Frontiers in oncology
Avec: Daniela Tomaselli , Clemens Steegborn , Antonello Mai ,

H19-Dependent Transcriptional Regulation of β3 and β4 Integrins Upon Estrogen and Hypoxia Favors Metastatic Potential in Prostate Cancer.

International journal of molecular sciences
Avec: Lorenza Bacci , Aurora Aiello , Cristian Ripoli , Rossella Loria , Dario Pugliese , Francesco Pierconti , Lidia Strigari , Francesco Pinto , Pier Francesco Bassi , Antonello Mai , Claudio Grassi , Alfredo Pontecorvi , Rita Falcioni , Antonella Farsetti , Simona Nanni

Effects of Glutathione Transferase-Targeting Nitrobenzoxadiazole Compounds in Relation to PD-L1 Status in Human Melanoma Cells.

Chemotherapy
Avec: Francesca Sciarretta , Chiara Fulci , Camilla Palumbo , Lucio Tentori , Grazia Graziani , Anna Maria Caccuri

Effect of α-Methoxy Substitution on the Anti-HIV Activity of Dihydropyrimidin-4(3 H)-ones.

Journal of medicinal chemistry
Avec: Maxim B Nawrozkij , Mariantonietta Forgione , Alexandre S Yablokov , Alessia Lucidi , Daniela Tomaselli , Alexandros Patsilinakos , Cristina Panella , Gebremedhin S Hailu , Ivan A Kirillov , Roger Badia , Eva Riveira-Muñoz , Emmanuele Crespan , Jorge I Armijos Rivera , Roberto Cirilli , Rino Ragno , José A Esté , Giovanni Maga , Antonello Mai ,

Current radiopharmaceuticals
Avec: Teresa Scotognella , Daria Maccora , Isabella Bruno , Marco Chinol , Massimo Castagnola , Francesco Collamati , Carlo Mancini-Terraciano , Silvio Morganti , Valerio Bocci , Elena Solfaroli Camillocci , Antonella Cartoni , Ilaria Fratoddi , Federica Marini , Iole Venditti , Riccardo Faccini , Alessandro Giordano

Radioguided surgery with β

Scientific reports
Avec: Francesco Collamati , Daria Maccora , Sergio Alfieri , Valerio Bocci , Antonella Cartoni , Angela Collarino , Micol De Simoni , Marta Fischetti , Ilaria Fratoddi , Alessandro Giordano , Carlo Mancini-Terracciano , Riccardo Mirabelli , Silvio Morganti , Giuseppe Quero , Teresa Scotognella , Elena Solfaroli Camillocci , Giacomo Traini , Iole Venditti , Riccardo Faccini

The Two-Faced Role of SIRT6 in Cancer.

Cancers
Avec: Francesco Fiorentino , Vincenzo Carafa , Gregorio Favale , Lucia Altucci , Antonello Mai ,

A potent HDAC inhibitor blocks Toxoplasma gondii tachyzoite growth and profoundly disrupts parasite gene expression.

International journal of antimicrobial agents
Avec: Thomas Mouveaux , Tom Boissavy , Emmanuel Roger , Christine Pierrot , Antonello Mai , Mathieu Gissot

Neuroprotective Effects of PARP Inhibitors in

Cells
Avec: Anna Maggiore , Assunta Maria Casale , Walter Toscanelli , Ugo Cappucci , Maddalena Grieco , Jean-Philippe Gagné , Guy G Poirier , Maria d'Erme , Lucia Piacentini

Simultaneous administration of EZH2 and BET inhibitors inhibits proliferation and clonogenic ability of metastatic prostate cancer cells.

Journal of enzyme inhibition and medicinal chemistry
Avec: Aide Negri , Marina Marozzi , Daniela Trisciuoglio , Antonello Mai , Federica Rizzi

METTL3 from Target Validation to the First Small-Molecule Inhibitors: A Medicinal Chemistry Journey.

Journal of medicinal chemistry
Avec: Francesco Fiorentino , Martina Menna , Sergio Valente , Antonello Mai

First-in-Class Selective Inhibitors of the Lysine Acetyltransferase KAT8.

Journal of medicinal chemistry
Avec: Francesco Fiorentino , Sara Sementilli , Martina Menna , Federica Turrisi , Stefano Tomassi , Francesca Romana Pellegrini , Angela Iuzzolino , Francesca D'Acunzo , Alessandra Feoli , Hannah Wapenaar , Sophie Taraglio , Caterina Fraschetti , Donatella Del Bufalo , Gianluca Sbardella , Frank J Dekker , Alessandro Paiardini , Daniela Trisciuoglio , Antonello Mai ,

Novel 1,4-Dihydropyridines as Specific Binders and Activators of SIRT3 Impair Cell Viability and Clonogenicity and Downregulate Hypoxia-Induced Targets in Cancer Cells.

Journal of medicinal chemistry
Avec: Clemens Zwergel , Michele Aventaggiato , Sabrina Garbo , Elisabetta Di Bello , Bruno Fassari , Beatrice Noce , Carola Castiello , Chiara Lambona , Federica Barreca , Rossella Fioravanti , Thomas Schmalz , Michael Weyand , Amelie Niedermeier , Marco Tripodi , Gianni Colotti , Clemens Steegborn , Cecilia Battistelli , Marco Tafani , Sergio Valente , Antonello Mai

Hydroxamate-based compounds are potent inhibitors of

Antimicrobial agents and chemotherapy
Avec: Tom Boissavy , Thomas Mouveaux , Emmanuel Roger , El Moukthar Aliouat , Christine Pierrot , Sergio Valente , Antonello Mai , Mathieu Gissot

BET Protein Inhibitor JQ1 Ameliorates Experimental Peritoneal Damage by Inhibition of Inflammation and Oxidative Stress.

Antioxidants (Basel, Switzerland)
Avec: Vanessa Marchant , Flavia Trionfetti , Lucia Tejedor-Santamaria , Sandra Rayego-Mateos , Giulio Bontempi , Alessandro Domenici , Paolo Menè , Antonello Mai , Catalina Martín-Cleary , Alberto Ortiz , Adrian M Ramos , Raffaele Strippoli , Marta Ruiz-Ortega

M

Nature communications
Avec: Gaia Di Timoteo , Andrea Giuliani , Adriano Setti , Martina C Biagi , Michela Lisi , Tiziana Santini , Alessia Grandioso , Davide Mariani , Francesco Castagnetti , Eleonora Perego , Sabrina Zappone , Serena Lattante , Mario Sabatelli , Giuseppe Vicidomini , Irene Bozzoni

Identification of Inhibitors to

International journal of molecular sciences
Avec: Tanira Matutino Bastos , Milena Botelho Pereira Soares , Caio Haddad Franco , Laura Alcântara , Lorenzo Antonini , Manuela Sabatino , Nicola Mautone , Lucio Holanda Freitas-Junior , Carolina Borsoi Moraes , Rino Ragno , Sergio Schenkman , Antonello Mai , Nilmar Silvio Moretti

From PARP1 to TNKS2 Inhibition: A Structure-Based Approach.

ACS medicinal chemistry letters
Avec: Stefano Tomassi , Julian Pfahler , Nicola Mautone , Annarita Rovere , Chiara Esposito , Daniela Passeri , Roberto Pellicciari , Ettore Novellino , Martin Pannek , Clemens Steegborn , Alessandro Paiardini , Antonello Mai ,

Characterization of water-soluble esters of nitrobenzoxadiazole-based GSTP1-1 inhibitors for cancer treatment.

Biochemical pharmacology
Avec: Veronica Di Paolo , Chiara Fulci , Anastasia De Luca , Stefano Tomassi , Massimo Serra , Manuel Scimeca , Cristina Geroni , Luigi Quintieri , Anna Maria Caccuri

Synthesis and characterisation of a new benzamide-containing nitrobenzoxadiazole as a GSTP1-1 inhibitor endowed with high stability to metabolic hydrolysis.

Journal of enzyme inhibition and medicinal chemistry
Avec: Veronica Di Paolo , Chiara Fulci , Francesca Sciarretta , Alessia Lucidi , Blasco Morozzo Della Rocca , Anastasia De Luca , Antonio Rosato , Luigi Quintieri , Anna Maria Caccuri

Tranylcypromine-Based LSD1 Inhibitors: Structure-Activity Relationships, Antiproliferative Effects in Leukemia, and Gene Target Modulation.

ChemMedChem
Avec: Rossella Fioravanti , Annalisa Romanelli , Nicola Mautone , Elisabetta Di Bello , Annarita Rovere , Davide Corinti , Clemens Zwergel , Sergio Valente , Oronza A Botrugno , Paola Dessanti , Stefania Vultaggio , Paola Vianello , Anna Cappa , Claudia Binda , Andrea Mattevi , Saverio Minucci , Ciro Mercurio , Mario Varasi , Antonello Mai

CDK9 as a Valuable Target in Cancer: From Natural Compounds Inhibitors to Current Treatment in Pediatric Soft Tissue Sarcomas.

Frontiers in pharmacology
Avec: Matteo Cassandri , Rossella Fioravanti , Silvia Pomella , Sergio Valente , Giada Del Baldo , Biagio De Angelis , Rossella Rota , Antonello Mai

Enzymatic and Biological Characterization of Novel Sirtuin Modulators against Cancer.

International journal of molecular sciences
Avec: Vincenzo Carafa , Angelita Poziello , Laura Della Torre , Pia Giovannelli , Marzia Di Donato , Elham Safadeh , Zhijun Yu , Alfonso Baldi , Gabriella Castoria , Daniela Tomaselli , Antonello Mai , Angela Nebbioso , Lucia Altucci

α,γ-Diketocarboxylic Acids and Their Esters Act as Carbonic Anhydrase IX and XII Selective Inhibitors.

ACS medicinal chemistry letters
Avec: Alessio Nocentini , Alessia Lucidi , Francesca Perut , Annamaria Massa , Daniela Tomaselli , Paola Gratteri , Nicola Baldini , Antonello Mai , Claudiu T Supuran

Anti-influenza A virus activity and structure-activity relationship of a series of nitrobenzoxadiazole derivatives.

Journal of enzyme inhibition and medicinal chemistry
Avec: Francesco Fiorentino , Marta De Angelis , Martina Menna , Annarita Rovere , Anna Maria Caccuri , Francesca D'Acunzo , Anna Teresa Palamara , Lucia Nencioni , Antonello Mai

SIRT5 Inhibition Induces Brown Fat-Like Phenotype in 3T3-L1 Preadipocytes.

Cells
Avec: Francesca Molinari , Alessandra Feraco , Simone Mirabilii , Serena Saladini , Luigi Sansone , Enza Vernucci , Giada Tomaselli , Vincenzo Marzolla , Matteo A Russo , Maria Rosaria Ricciardi , Agostino Tafuri , Antonello Mai , Massimiliano Caprio , Marco Tafani , Andrea Armani

Transcriptomic and genomic studies classify NKL54 as a histone deacetylase inhibitor with indirect influence on MEF2-dependent transcription.

Nucleic acids research
Avec: Martina Minisini , Eros Di Giorgio , Emanuela Kerschbamer , Emiliano Dalla , Massimo Faggiani , Elisa Franforte , Franz-Josef Meyer-Almes , Rino Ragno , Lorenzo Antonini , Antonello Mai , Francesco Fiorentino , Monica Chinellato , Stefano Perin , Laura Cendron , Christian X Weichenberger , Alessandro Angelini , Claudio Brancolini

HDAC1-3 inhibition increases SARS-CoV-2 replication and productive infection in lung mesothelial and epithelial cells.

Frontiers in cellular and infection microbiology
Avec: Flavia Trionfetti , Tonino Alonzi , Giulio Bontempi , Michela Terri , Cecilia Battistelli , Claudia Montaldo , Federica Repele , Sergio Valente , Clemens Zwergel , Giulia Matusali , Fabrizio Maggi , Delia Goletti , Marco Tripodi , Antonello Mai , Raffaele Strippoli

Specific Inhibitors of Mitochondrial Deacylase Sirtuin 4 Endowed with Cellular Activity.

Journal of medicinal chemistry
Avec: Martin Pannek , Zayan Alhalabi , Daniela Tomaselli , Martina Menna , Francesco Fiorentino , Dina Robaa , Michael Weyand , Maximilian Puhlmann , Stefano Tomassi , Federica Barreca , Marco Tafani , Elma Zaganjor , Marcia C Haigis , Wolfgang Sippl , Antonello Mai , Clemens Steegborn

Réseau de co-auteurs

Antonello Mai 54 collaborations
Francesco Fiorentino 19 collaborations
Sergio Valente 11 collaborations
Daniela Tomaselli 8 collaborations
Nicola Mautone 8 collaborations
Alessia Lucidi 7 collaborations
Lucia Altucci 7 collaborations
Martina Menna 7 collaborations
Clemens Steegborn 6 collaborations
Marco Tafani 5 collaborations
Anna Maria Caccuri 5 collaborations
Daniela Trisciuoglio 5 collaborations
Vincenzo Carafa 5 collaborations
Rino Ragno 5 collaborations
Stefano Tomassi 5 collaborations
Rossella Fioravanti 4 collaborations
Annarita Rovere 4 collaborations
Emanuele Fabbrizi 4 collaborations
Clemens Zwergel 4 collaborations
Christine Pierrot 3 collaborations
Rosaria Benedetti 3 collaborations
Tommaso De Marchi 3 collaborations
Emma Niméus 3 collaborations
Chiara Papulino 3 collaborations
Ugo Chianese 3 collaborations
Angela Nebbioso 3 collaborations
Veronica Di Paolo 3 collaborations
Luigi Quintieri 3 collaborations
Francesca Romana Pellegrini 3 collaborations
Lorenzo Antonini 3 collaborations
Donatella Del Bufalo 3 collaborations
Francesca D'Acunzo 3 collaborations
Gianluca Sbardella 3 collaborations
Jujun Zhou 3 collaborations
John R Horton 3 collaborations
Ren Ren 3 collaborations
Robert M Blumenthal 3 collaborations
Xing Zhang 3 collaborations
Xiaodong Cheng 3 collaborations
Valerio Bocci 3 collaborations
Riccardo Faccini 3 collaborations
Alessandro Paiardini 3 collaborations
Federica Barreca 3 collaborations
Chiara Fulci 3 collaborations
Julien Lancelot 2 collaborations
Raymond J Pierce 2 collaborations
Johan Schultz 2 collaborations
Carmela Dell'Aversana 2 collaborations
Alfonso Baldi 2 collaborations
Francesco Iovino 2 collaborations
Enza Vernucci 2 collaborations
Angela Iuzzolino 2 collaborations
Mohammad Salik Zeya Ansari 2 collaborations
Manuela Sabatino 2 collaborations
Daniela Passeri 2 collaborations
Roberto Pellicciari 2 collaborations
Alessia Ciogli 2 collaborations
Monica Viviano 2 collaborations
Alessandra Feoli 2 collaborations
Milan Mladenović 2 collaborations
Alessio Nocentini 2 collaborations
Claudiu T Supuran 2 collaborations
Laura Della Torre 2 collaborations
Giulia Sgueglia 2 collaborations
Marzia Di Donato 2 collaborations
Frank J Dekker 2 collaborations
Dina Robaa 2 collaborations
Wolfgang Sippl 2 collaborations
Carlo Mancini-Terracciano 2 collaborations
Matteo Cassandri 2 collaborations
Silvia Pomella 2 collaborations
Rossella Rota 2 collaborations
Saverio Minucci 2 collaborations
Andrea Mattevi 2 collaborations
Michele Aventaggiato 2 collaborations
Luigi Sansone 2 collaborations
Matteo A Russo 2 collaborations
Qin Chen 2 collaborations
Jie Yang 2 collaborations
Bigang Liu 2 collaborations
Caleb Chang 2 collaborations
Chuxuan Li 2 collaborations
Leora Maksoud 2 collaborations
Yifei Yang 2 collaborations
Taiping Chen 2 collaborations
Yang Gao 2 collaborations
Francesco Pierconti 2 collaborations
Francesco Pinto 2 collaborations
Claudio Grassi 2 collaborations
Alfredo Pontecorvi 2 collaborations
Lidia Strigari 2 collaborations
Antonella Farsetti 2 collaborations
Simona Nanni 2 collaborations
Francesca Sciarretta 2 collaborations
Teresa Scotognella 2 collaborations
Daria Maccora 2 collaborations
Francesco Collamati 2 collaborations
Silvio Morganti 2 collaborations
Elena Solfaroli Camillocci 2 collaborations
Antonella Cartoni 2 collaborations
Ilaria Fratoddi 2 collaborations
Iole Venditti 2 collaborations
Alessandro Giordano 2 collaborations
Thomas Mouveaux 2 collaborations
Tom Boissavy 2 collaborations
Emmanuel Roger 2 collaborations
Mathieu Gissot 2 collaborations
Elisabetta Di Bello 2 collaborations
Michael Weyand 2 collaborations
Marco Tripodi 2 collaborations
Cecilia Battistelli 2 collaborations
Flavia Trionfetti 2 collaborations
Giulio Bontempi 2 collaborations
Raffaele Strippoli 2 collaborations
Martin Pannek 2 collaborations
Anastasia De Luca 2 collaborations
Daria Monaldi 1 collaboration
Martin Marek 1 collaboration
Nathalie Wössner 1 collaboration
Elizabeth Ramos-Morales 1 collaboration
Christophe Romier 1 collaboration
Manfred Jung 1 collaboration
Anne Bouchut 1 collaboration
Sophia Lafitte 1 collaboration
Urban Hoglund 1 collaboration
Roberta Mazzone 1 collaboration
Giancarlo Fabrizi 1 collaboration
Dany Pechalrieu 1 collaboration
Paola B Arimondo 1 collaboration
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